PLD Inhibitor, FIPI

A potent phospholipase D inhibitor

Cat. No.: AUR10283

CAS Number: 939055-18-2

Documents:

SizePrice

50 mg

$ 725

Tags FIPI PLD inhibitor phospholipase D inhiibitor CAS#939055-18-2 939055-18-2 Auroramedbiochem

Alternate Names

Appearance

Off-white solid

Formulation

N/A

CAS Number

939055-18-2

Molecular Formula

C23H24FN5O2

Molecular Weight

421.48

Purity

≥98% by HPLC

Solubility

DMSO (100 mg/ml)

Handling

Protect from air and light

Country of origin

USA

Storage temperature

+2 to +8 ◦C

Shipping Condition

Shelf life

24 months

MDL number

MFCD18382115

PubChem CID

16739265

SMILES

C1CN(CCC1N2C3=CC=CC=C3NC2=O)CCNC(=O)C4=CC5=C(N4)C=CC(=C5)F

InChI

InChI=1S/C23H24FN5O2/c24-16-5-6-18-15(13-16)14-20(26-18)22(30)25-9-12-28-10-7-17(8-11-28)29-21-4-2-1-3-19(21)27-23(29)31/h1-6,13-14,17,26H,7-12H2,(H,25,30)(H,27,31)

InChI key

LHABRXRGDLASIH-UHFFFAOYSA-N

FIPI (5-Fluoro-2-indolyl deschlorohalopemide), a derivative of halopemide, is a potent and selective inhibitor of phospholipase D with IC50 of 25 nM and 20 nM for PLD1 and PLD2, respectively.